SCHEMBL8934929

SCHEMBL8934929

O=C(c1ccc(-c2ccc(O)cc2)cc1)N1CCNCC1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.64
MKNK1 Q9BUB5 2/20 0.62
MKNK2 Q9HBH9 2/20 0.62
HPGD P15428 3/20 0.58
CCNC P24863 7/20 0.57
CDK8 P49336 7/20 0.57
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
MAPK1 P28482 1/20 0.53
RIPK1 Q13546 1/20 0.50
TDO2 P48775 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4505138 0.95 SIGMAR1 (0.70) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL8260488 0.93 SIGMAR1 (0.72) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL8358137 0.87 SIGMAR1 (0.81) SIGMAR1MKNK1MKNK2HPGDL3MBTL1
SCHEMBL5266293 0.86 SIGMAR1 (0.80) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL16574186 0.85 GABRD (0.66) SIGMAR1MKNK1MKNK2HPGDCCNC
Hydrochloric Acid SCHEMBL4763940 0.85 SIGMAR1 (0.77) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL29800584 0.85 SIGMAR1 (0.62) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL7425708 0.83 MKNK1 (0.72) SIGMAR1MKNK1MKNK2HPGDCCNC
SCHEMBL3583338 0.82 HPGD (0.73) SIGMAR1MKNK1MKNK2HPGDL3MBTL1
SCHEMBL14523155 0.81 HPGD (0.64) HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
WO-2022149617-A1 COMPOUND LIBRARY 中外製薬株式会社 2022-07-14 WO disclosed
WO-1996029088-A1 NOVEL PIPERAZINE DERIVATIVES AS TYPE IL-1 RECEPTOR ANTAGONISTS AFFYMAX TECHNOLOGIES N.V. (AN) 1996-09-26 WO disclosed