SCHEMBL8935316

SCHEMBL8935316

C[C@H](NCc1ccc(OCc2ccccc2)cc1)C(=O)N(C)C

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.57
MAOB P27338 3/20 0.55
SCN9A Q15858 2/20 0.55
MAOA P21397 1/20 0.55
ALOX5 P09917 1/20 0.54
LTA4H P09960 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394431 1.00 BCHE (0.57) BCHEMAOBSCN9AMAOAALOX5
SCHEMBL2493421 0.86 SIGMAR1 (0.49)
SCHEMBL9129586 0.86 MAOB (0.76) MAOBSCN9AMAOA
SCHEMBL8935307 0.86 ALOX5 (0.60) MAOBSCN9AMAOAALOX5
SCHEMBL963148 0.86 MAOB (0.76) MAOBSCN9AMAOA
SCHEMBL15479186 0.85 BCHE (0.61) BCHEMAOBSCN9AMAOA
SCHEMBL8935359 0.85 MMP9 (0.56) BCHEMAOBALOX5
SCHEMBL8935334 0.85 MMP9 (0.56) BCHEMAOBALOX5
SCHEMBL7397586 0.84 MAOB (0.57) MAOBSCN9AMAOA
SCHEMBL965367 0.84 SCN9A (0.76) MAOBSCN9AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502079-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS FARMITALIA CARLO ERBA S.R.L. (IT) 1996-03-26 US disclosed
US-5484879-A AROMATIC DIAMINES SUBSTITUTED WITH TRIFLUOROMETHYL GROUPS OCCIDENTAL CHEMICAL CORPORATION (US) 1996-01-16 US disclosed
US-5391577-A Active on central nervous system; antiepileptic agents FARMITALIA CARLO ERBA S R L (IT) 1995-02-21 US disclosed
US-5236957-A Antiepileptic agents FARMITALIA CARLO ERBA SRL (IT) 1993-08-17 US disclosed