SCHEMBL8935817

SCHEMBL8935817

O=C1c2ccccc2C(=O)N1CC(CCc1ccccc1)OS(=O)(=O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.48
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
BLM P54132 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 3/20 0.38
ALDH2 P05091 2/20 0.38
ALDH3A1 P30838 2/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
PARK7 Q99497 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935885 0.83 MAPK1 (0.58) CASP3MAPK1TDP1L3MBTL1CA1
SCHEMBL19285727 0.73 CASP3 (0.58) CASP3MAPK1TDP1L3MBTL1BLM
SCHEMBL21981027 0.73 BLM (0.41) BLMCA1CA2ALDH1A1KDM4E
SCHEMBL19737275 0.71 CASP3 (0.55) CASP3MAPK1TDP1L3MBTL1BLM
SCHEMBL1059677 0.70 CASP3 (0.58) CASP3TDP1L3MBTL1BLMCA1
SCHEMBL25467952 0.69 ALDH1A1 (0.37) CASP3MAPK1ALDH1A1MAPTRAB9A
SCHEMBL6515182 0.69 PPARG (0.50) BLM
SCHEMBL7425913 0.69 PPARG (0.50) BLM
SCHEMBL15956280 0.68 TDP1 (0.56) CASP3MAPK1TDP1L3MBTL1CA1
SCHEMBL290900 0.67 RAB9A (0.50) CASP3TDP1L3MBTL1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5531978-A CHELATE COMPOUNDS, IMAGING NYCOMED IMAGING AS (NO) 1996-07-02 US disclosed
US-5419893-A Aminopolycarboxylic acids and derivatives thereof for magnetic resonance imaging NYCOMED IMAGING AS (NO) 1995-05-30 US disclosed
US-5198208-A Chelate compounds for diagnosis by magnetic resonance imaging, ultrasound or radiation therapy NYCOMED IMAGING AS (NO) 1993-03-30 US disclosed
EP-0466200-A1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1992-01-15 EP disclosed
WO-1989000557-A1 AMINOPOLYCARBOXYLIC ACIDS AND DERIVATIVES THEREOF COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1989-01-26 WO disclosed