SCHEMBL8936121

SCHEMBL8936121

CC(Cl)CN(CC#N)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.47
ALDH1A1 P00352 4/20 0.42
CYP1A2 P05177 2/20 0.40
MAPK1 P28482 1/20 0.40
TSHR P16473 4/20 0.38
LMNA P02545 3/20 0.38
CYP3A4 P08684 2/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRK1 P41145 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
USP2 O75604 1/20 0.38
MAOA P21397 1/20 0.38
PYCR1 P32322 1/20 0.38
CTSB P07858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936116 1.00 MAOB (0.47) MAOBALDH1A1CYP1A2MAPK1TSHR
SCHEMBL17986869 0.84 MAOB (0.42) MAOBALDH1A1CYP1A2MAPK1TSHR
SCHEMBL31228482 0.83 ALDH1A1 (0.41) MAOBALDH1A1CYP1A2MAPK1TSHR
SCHEMBL27968570 0.80 ALDH1A1 (0.56) MAOBALDH1A1CYP1A2TSHRLMNA
SCHEMBL8986000 0.77 OPRK1 (0.49) ALDH1A1CYP1A2SLC6A2SLC6A4ADRA1A
SCHEMBL12265182 0.77 TSHR (0.47) ALDH1A1CYP1A2TSHRLMNACYP3A4
Hydrochloric Acid SCHEMBL31094860 0.75 ALDH1A1 (0.48) ALDH1A1CYP1A2MAPK1TSHRLMNA
SCHEMBL5703569 0.75 NR1D1 (0.53) MAOBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL20135644 0.74 MEN1 (0.45) TSHRLMNARECQLMEN1KMT2A
SCHEMBL20135643 0.74 MEN1 (0.45) TSHRLMNARECQLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659178-A4 CHIRAL QUINOLONE INTERMEDIATES. ABBOTT LAB (US) 1996-03-27 EP disclosed
EP-0659178-A1 CHIRAL QUINOLONE INTERMEDIATES ABBOTT LABORATORIES (US) 1995-06-28 EP disclosed
WO-1994006766-A1 CHIRAL QUINOLONE INTERMEDIATES ABBOTT LABORATORIES (US) 1994-03-31 WO disclosed
US-5252747-A Chiral quinolone intermediates ABBOTT LABORATORIES (US) 1993-10-12 US disclosed