SCHEMBL8939741

SCHEMBL8939741

[c]1ccc(Cc2cccc(Oc3ccccc3)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 4/20 0.44
HTT P42858 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SRD5A2 P31213 1/20 0.44
MAOB P27338 1/20 0.43
P2RX3 P56373 1/20 0.42
IDH1 O75874 1/20 0.42
FDFT1 P37268 1/20 0.41
TSHR P16473 2/20 0.41
LTA4H P09960 1/20 0.41
CALM1 P0DP23 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPV6 Q9H1D0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23312282 0.87 ALDH1A1 (0.50) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL8896665 0.87 TSHR (0.55) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL22550294 0.87 CALM1 (0.55) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL9816693 0.85 SRD5A2 (0.58) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL6978760 0.81 CHRM2 (0.53) MAOBLTA4H
Ethylene Glycol SCHEMBL28545403 0.80 TSHR (0.51) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL27630414 0.79 LTA4H (0.57) KDM4EALDH1A1HTTSMN1; SMN2SRD5A2
SCHEMBL79755 0.79 CALM1 (0.67) KDM4EALDH1A1IDH1TSHRLTA4H
SCHEMBL921840 0.77 ALDH1A1 (0.45) KDM4EALDH1A1HTTTDP1HPGD
SCHEMBL8939739 0.77 KDM4E (0.42) KDM4EALDH1A1HTTTDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516797-A SUPPRESSING GRAFT REJECTION VERTEX PHARMACEUTICALS, INCORPORATED (US) 1996-05-14 US disclosed
US-5330993-A Immunosuppressive compounds VERTEX PHARMACEUTICALS, INC. (US) 1994-07-19 US disclosed