SCHEMBL8939773

SCHEMBL8939773

COc1c[c]c(Cc2ccc(-c3ccccc3)cc2)c(OC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
HPGD P15428 3/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TUBB4A P04350 4/20 0.39
TUBB P07437 4/20 0.39
TUBA3C P0DPH7 4/20 0.39
TUBA1B P68363 4/20 0.39
TUBA4A P68366 4/20 0.39
TUBB4B P68371 4/20 0.39
TUBB3 Q13509 4/20 0.39
TUBB2A Q13885 4/20 0.39
TUBB8 Q3ZCM7 4/20 0.39
TUBA3E Q6PEY2 4/20 0.39
TUBA1A Q71U36 4/20 0.39
TUBA1C Q9BQE3 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939769 0.91 LTA4H (0.42) KDM4EMAPTHPGDALDH1A1TUBB4A
SCHEMBL8939758 0.82 APP (0.41) ALDH1A1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL6160386 0.77 ABCB1 (0.44) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8190525 0.77 MEN1 (0.47) KDM4EKMT2AALDH1A1TDP1MEN1
SCHEMBL8827586 0.76 HTR7 (0.40) PDE4BPDE4D
SCHEMBL7429582 0.75 BCHE (0.40) HPGD
SCHEMBL7746427 0.75 HTR2A (0.42) HPGD
SCHEMBL6161069 0.74 ALDH1A1 (0.42) KDM4EHPGDKMT2AALDH1A1LMNA
SCHEMBL7746382 0.73 TDP1 (0.40) HPGDTDP1L3MBTL1
SCHEMBL8939724 0.73 MAOB (0.44) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516797-A SUPPRESSING GRAFT REJECTION VERTEX PHARMACEUTICALS, INCORPORATED (US) 1996-05-14 US disclosed
US-5330993-A Immunosuppressive compounds VERTEX PHARMACEUTICALS, INC. (US) 1994-07-19 US disclosed