SCHEMBL8939781

SCHEMBL8939781

Fc1cc[c]c(Cc2ccccc2)c1F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.41
HTR2A P28223 2/20 0.33
ALOX5 P09917 1/20 0.32
BCL2 P10415 1/20 0.31
BCL2L1 Q07817 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
CYP2A6 P11509 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
LTA4H P09960 2/20 0.31
ALDH1A1 P00352 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106395 0.83 CALM1 (0.39) CALM1HTR2AALOX5BCL2BCL2L1
SCHEMBL16798254 0.81 CALM1 (0.38) CALM1ALOX5ALDH1A1
SCHEMBL8859945 0.80 CALM1 (0.37) CALM1HTR2ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL7459473 0.78 CALM1 (0.42) CALM1HTR2AALOX5BCL2BCL2L1
SCHEMBL8466360 0.77 CALM1 (0.55) CALM1HTR2ABCL2BCL2L1TAAR1
SCHEMBL455831 0.71
SCHEMBL20487629 0.71 LOXL2 (0.31) LOXL2
SCHEMBL20486385 0.71
SCHEMBL20487021 0.71 PRMT6 (0.31) KDM4E
SCHEMBL8802600 0.69 BCL2 (0.44) CALM1ALOX5BCL2BCL2L1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516797-A SUPPRESSING GRAFT REJECTION VERTEX PHARMACEUTICALS, INCORPORATED (US) 1996-05-14 US disclosed
US-5330993-A Immunosuppressive compounds VERTEX PHARMACEUTICALS, INC. (US) 1994-07-19 US disclosed