SCHEMBL8945917

SCHEMBL8945917

CNC(Cc1ccccc1N)c1ncc(C)s1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
CACNA2D1 P54289 1/20 0.33
CTSA P10619 1/20 0.32
KDR P35968 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945905 0.85 YTHDC1 (0.33) KDR
SCHEMBL8945855 0.78 HDAC1 (0.35) SLC6A3HDAC1
SCHEMBL8945778 0.77 SLC6A2 (0.37)
SCHEMBL8945765 0.76 CYP3A4 (0.33) SLC6A3KMT2A
SCHEMBL8945988 0.72 YTHDC1 (0.33) SLC6A3KMT2A
SCHEMBL8945955 0.71 TSHR (0.38) SLC6A3
SCHEMBL4542976 0.71 GUCY1B2 (0.39) NOS1SLC6A3CACNA2D1CTSA
SCHEMBL9001661 0.71 ALDH1A1 (0.42)
SCHEMBL8946109 0.71 YTHDC1 (0.32) HDAC3HDAC1
SCHEMBL8946102 0.71 SLC6A2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed