SCHEMBL8945923

SCHEMBL8945923

CN1C(c2ccccc2)=Nc2ccccc2CC1c1ccsc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.35
DRD2 P14416 3/20 0.33
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
CYP2E1 P05181 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2B6 P20813 1/20 0.31
EGFR P00533 1/20 0.31
GBA1 P04062 1/20 0.30
CCR3 P51677 1/20 0.30
HTR1A P08908 1/20 0.30
HTR7 P34969 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945921 0.99 HRH4 (0.34) HRH4DRD2MAOAMAOBCYP2E1
SCHEMBL8945994 0.84 HSD17B10 (0.34) HRH4
SCHEMBL8946148 0.81 ADORA2B (0.33) HRH4
SCHEMBL8945925 0.81 ADORA2B (0.32) HRH4
Hydrochloric Acid SCHEMBL8945865 0.80 ADORA2B (0.32)
SCHEMBL8945861 0.79 SMN1; SMN2 (0.32)
Hydrochloric Acid SCHEMBL8945951 0.79 ADORA2B (0.31)
SCHEMBL8946123 0.78 OPRM1 (0.31) DRD2
SCHEMBL8945967 0.77 HRH4 (0.34) HRH4DRD2MAOAMAOBEGFR
Hydrochloric Acid SCHEMBL8945756 0.76 HRH4 (0.34) HRH4DRD2MAOAMAOBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed