SCHEMBL8946148

SCHEMBL8946148

CCC1=Nc2ccccc2CC(c2ccsc2)N1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
OPRM1 P35372 3/20 0.31
OPRD1 P41143 2/20 0.31
OPRK1 P41145 2/20 0.31
SIRT3 Q9NTG7 1/20 0.31
SIRT5 Q9NXA8 1/20 0.31
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945865 0.99 ADORA2B (0.32) ADORA2BSMN1; SMN2LMNAOPRM1OPRD1
SCHEMBL8945861 0.91 SMN1; SMN2 (0.32) ADORA2BSMN1; SMN2LMNAMEN1HTT
SCHEMBL8946123 0.87 OPRM1 (0.31) ADORA2BOPRM1OPRD1OPRK1MEN1
SCHEMBL11270824 0.84 CHRNB2 (0.37) LMNAMEN1KMT2AALDH1A1GAA
SCHEMBL8945994 0.84 HSD17B10 (0.34) ADORA2BSMN1; SMN2LMNASIRT3SIRT5
SCHEMBL8946144 0.81 CYP19A1 (0.34) KMT2AHRH4
SCHEMBL9583461 0.81 MAOA (0.40) LMNAMEN1KMT2AHPGD
SCHEMBL8945923 0.81 HRH4 (0.35) HRH4
SCHEMBL8945925 0.81 ADORA2B (0.32) ADORA2BOPRM1OPRK1HRH4
SCHEMBL9584219 0.80 MAOB (0.41) LMNAMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed