SCHEMBL8946052

SCHEMBL8946052

CC1=Nc2ccccc2CC(c2ccccn2)N1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
NPEPPS P55786 3/20 0.39
CXCR4 P61073 4/20 0.37
RIPK1 Q13546 1/20 0.35
DRD2 P14416 1/20 0.35
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
CASP1 P29466 2/20 0.34
GFER P55789 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
CASP7 P55210 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP2D6 P10635 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8945879 0.99 ALDH1A1 (0.39) ALDH1A1MAPTNPEPPSCXCR4RIPK1
Water SCHEMBL8945872 0.99 ALDH1A1 (0.39) ALDH1A1MAPTNPEPPSCXCR4RIPK1
SCHEMBL8946051 0.84 NPEPPS (0.37) ALDH1A1MAPTNPEPPSCXCR4RIPK1
SCHEMBL8946119 0.83 NPEPPS (0.39) ALDH1A1MAPTNPEPPSCXCR4RIPK1
Hydrochloric Acid SCHEMBL8946103 0.82 NPEPPS (0.36) ALDH1A1MAPTNPEPPSCXCR4RIPK1
Hydrochloric Acid SCHEMBL8945986 0.82 NPEPPS (0.36) ALDH1A1MAPTNPEPPSCXCR4RIPK1
Hydrochloric Acid SCHEMBL8945945 0.81 NPEPPS (0.38) ALDH1A1MAPTNPEPPSCXCR4RIPK1
Dazepinil SCHEMBL499286 0.80 CHRNB2 (0.40) RIPK1CYP2D6MEN1RECQLKMT2A
SCHEMBL8945898 0.79 CYP19A1 (0.35) DRD2L3MBTL1CYP2D6MEN1RECQL
SCHEMBL11266015 0.77 MAOA (0.43) HPGDCYP2D6MEN1RECQLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed