SCHEMBL8946919

SCHEMBL8946919

COc1ccc2[nH]c(I)c(CCNC(=O)C3CC3)c2c1

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 13/20 0.78
MTNR1B P49286 12/20 0.78
CYP1A2 P05177 2/20 0.74
CYP3A4 P08684 1/20 0.74
CYP2D6 P10635 1/20 0.74
CYP2C9 P11712 1/20 0.74
NQO2 P16083 1/20 0.74
TSHR P16473 1/20 0.74
CYP2C19 P33261 1/20 0.74
ALDH1A1 P00352 3/20 0.70
KDM4E B2RXH2 1/20 0.59
HSD17B10 Q99714 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946895 0.88 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2ALDH1A1KDM4E
SCHEMBL8946906 0.87 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2ALDH1A1KDM4E
SCHEMBL8946963 0.85 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
Iodomelatonin SCHEMBL163451 0.85 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8947176 0.85 MTNR1B (1.00) MTNR1AMTNR1BCYP1A2ALDH1A1KDM4E
SCHEMBL15428091 0.84 MTNR1A (0.74) MTNR1AMTNR1BCYP1A2NQO2ALDH1A1
SCHEMBL21075898 0.84 MTNR1A (0.92) MTNR1AMTNR1BALDH1A1KDM4EHSD17B10
SCHEMBL29409541 0.82 ALDH1A1 (0.80) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL4756887 0.82 ALDH1A1 (1.00) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL4759323 0.78 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552428-A ANTIARRHYTHMIA AGENTS FOR CARDIOVASCULAR DISORDERS USING MELATONIN DERIVATIVES INSTITUTO FARMACOLOGICO LOMBARDO-IFLO, S.A.S. (IT) 1996-09-03 US claimed
US-5552428-A ANTIARRHYTHMIA AGENTS FOR CARDIOVASCULAR DISORDERS USING MELATONIN DERIVATIVES INSTITUTO FARMACOLOGICO LOMBARDO-IFLO, S.A.S. (IT) 1996-09-03 US disclosed