SCHEMBL8946963

SCHEMBL8946963

COc1ccc2[nH]c(-c3ccccc3)c(CCNC(=O)C3CC3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 1.00
MTNR1B P49286 9/20 1.00
KDM4E B2RXH2 1/20 0.76
ALDH1A1 P00352 1/20 0.76
CYP1A2 P05177 1/20 0.76
CYP3A4 P08684 1/20 0.76
CYP2D6 P10635 1/20 0.76
CYP2C9 P11712 1/20 0.76
HPGD P15428 1/20 0.76
CYP2C19 P33261 1/20 0.76
HSD17B10 Q99714 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3508630 0.86 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL29759426 0.86 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL8946919 0.85 MTNR1A (0.78) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL13436463 0.85 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL8946895 0.84 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL8946906 0.83 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL8947176 0.82 MTNR1B (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL13436465 0.81 MTNR1A (0.88) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL15428091 0.81 MTNR1A (0.74) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL21075898 0.81 MTNR1A (0.92) MTNR1AMTNR1BKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552428-A ANTIARRHYTHMIA AGENTS FOR CARDIOVASCULAR DISORDERS USING MELATONIN DERIVATIVES INSTITUTO FARMACOLOGICO LOMBARDO-IFLO, S.A.S. (IT) 1996-09-03 US disclosed