SCHEMBL8947810

SCHEMBL8947810

Cc1cc2c(-c3ccccc3)c(CCNC(=O)OCc3ccccc3)n(C)c(=O)c2cc1C

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.53
L3MBTL1 Q9Y468 1/20 0.45
KAT2B Q92831 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DPP4 P27487 2/20 0.43
IDO1 P14902 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947918 0.77 TACR1 (0.52) TACR1LMNADPP4
SCHEMBL8785081 0.76 TACR1 (0.58) TACR1L3MBTL1LMNASMN1; SMN2
SCHEMBL8936490 0.74 TACR1 (0.73) TACR1
SCHEMBL8784483 0.74 TACR1 (0.56) TACR1DPP4
SCHEMBL8947993 0.74 DPP4 (0.71) TACR1DPP4
SCHEMBL8786372 0.74 TACR1 (0.51) TACR1DPP4
SCHEMBL5236388 0.72 DPP4 (0.70) TACR1DPP4
SCHEMBL8784402 0.71 KCNA5 (0.55) TACR1SMN1; SMN2DPP4
SCHEMBL8785655 0.71 TACR1 (0.56) TACR1LMNASMN1; SMN2HTT
Benzyl Phenethylcarbamate SCHEMBL4287199 0.69 LMNA (0.73) L3MBTL1LMNASMN1; SMN2IDO1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed