SCHEMBL8947894

SCHEMBL8947894

Cn1c(=O)oc2cc(CCCCN3CCC(C(=O)c4ccc(Cl)cc4)CC3)ccc21

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.56
HTR1A P08908 2/20 0.51
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
HTR2A P28223 1/20 0.48
LMNA P02545 1/20 0.47
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948109 0.91 HTR2A (0.61) HTR1AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8948004 0.91 HTR1A (0.58) KCNH2HTR1AKDM4ECYP1A2CYP3A4
SCHEMBL8948067 0.89 HTR1A (0.56) KCNH2HTR1AKDM4ECYP1A2CYP3A4
SCHEMBL8947961 0.82 LMNA (0.50) KCNH2HTR1AHTR2ALMNASLC6A2
SCHEMBL8947923 0.81 KCNH2 (0.56) KCNH2HTR1AKDM4ECYP1A2CYP3A4
SCHEMBL5655532 0.78 HTR1A (0.56) HTR1ASLC6A2SLC6A4SLC6A3TP53
SCHEMBL8947873 0.78 HTR2A (0.56) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL8870844 0.77 SIGMAR1 (0.66) HTR1ACYP1A2CYP3A4CYP2D6TP53
SCHEMBL8871026 0.76 SIGMAR1 (0.66) KCNH2HTR1ATP53
SCHEMBL8947902 0.76 KCNH2 (0.53) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed