SCHEMBL8948067

SCHEMBL8948067

COc1ccc(C(=O)C2CCN(CCCCc3ccc4c(c3)oc(=O)n4C)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.56
TSHR P16473 2/20 0.48
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
HTR2A P28223 1/20 0.47
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 1/20 0.46
KCNH2 Q12809 1/20 0.46
SLC18A3 Q16572 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947961 0.94 LMNA (0.50) HTR1ATSHRLMNASMN1; SMN2HTR2A
SCHEMBL8947894 0.89 KCNH2 (0.56) HTR1ALMNASMN1; SMN2KDM4ECYP1A2
SCHEMBL8948109 0.89 HTR2A (0.61) HTR1AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8948004 0.89 HTR1A (0.58) HTR1AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9161222 0.83 LMNA (0.47) TSHRLMNASMN1; SMN2KDM4ECYP1A2
SCHEMBL8947963 0.77 SIGMAR1 (0.50)
SCHEMBL8948008 0.77 HTR1A (0.57) HTR1ATSHRLMNASMN1; SMN2KDM4E
SCHEMBL8947957 0.77 HTR1A (0.65) HTR1AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL5655532 0.77 HTR1A (0.56) HTR1AALDH1A1MEN1KMT2A
SCHEMBL8947873 0.77 HTR2A (0.56) KDM4ECYP1A2CYP3A4CYP2D6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed