SCHEMBL8948007

SCHEMBL8948007

Cn1c(=O)sc2cc(CCN3CCC(C(=O)c4ccc(F)cc4)CC3)ccc21

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.66
HTR2C P28335 5/20 0.65
HTR2A P28223 3/20 0.65
HTR7 P34969 3/20 0.65
HTR6 P50406 3/20 0.65
SIGMAR1 Q99720 6/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948030 0.93 SIGMAR1 (0.62) HTR1AHTR2CHTR2AHTR7HTR6
SCHEMBL8947935 0.87 HTR2A (0.59) HTR1AHTR2CHTR2AHTR7HTR6
SCHEMBL8947974 0.85 SIGMAR1 (0.64) HTR2CHTR2AHTR7HTR6SIGMAR1
SCHEMBL8870940 0.84 SIGMAR1 (0.82) HTR1AHTR2CSIGMAR1
SCHEMBL8948011 0.84 HTR1A (0.60) HTR1AHTR2CHTR2AHTR7HTR6
SCHEMBL8948061 0.82 SIGMAR1 (0.52) HTR2CHTR2AHTR7HTR6SIGMAR1
SCHEMBL8948192 0.81 HTR1A (0.65) HTR1AHTR2CHTR2AHTR7
SCHEMBL8948078 0.81 HTR2A (0.55) HTR2CHTR2AHTR7HTR6SIGMAR1
SCHEMBL8947898 0.81 HTR2A (0.55) HTR2CHTR2AHTR7HTR6SIGMAR1
SCHEMBL8948202 0.81 HTR2C (0.67) HTR1AHTR2CHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed