SCHEMBL8947975

SCHEMBL8947975

O=C(c1ccccc1)C1CCN(CCn2c(=O)sc3ccccc32)CC1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
HTR2A P28223 1/20 0.55
HTT P42858 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
DRD2 P14416 1/20 0.54
DRD4 P21917 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948121 0.91 HTR2A (0.57) SIGMAR1HTR2ADRD2DRD4
SCHEMBL8948100 0.88 SIGMAR1 (0.48) SIGMAR1DRD2DRD4
SCHEMBL8947958 0.88 SMN1; SMN2 (0.55)
SCHEMBL8947939 0.86 DRD2 (0.53) SIGMAR1DRD2DRD4
SCHEMBL11707845 0.85 KDM4E (0.58) HTR2A
SCHEMBL8948053 0.84 TSHR (0.52) HTT
SCHEMBL8870364 0.82 SIGMAR1 (0.60) SIGMAR1DRD2DRD4
SCHEMBL3028533 0.80 DRD2 (0.60) DRD2DRD4
SCHEMBL8947787 0.80 SIGMAR1 (0.58) SIGMAR1HTR2A
SCHEMBL8870387 0.79 SIGMAR1 (0.61) SIGMAR1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed