SCHEMBL8870940

SCHEMBL8870940

Cn1c(=O)sc2cc(CCN3CCC(Cc4ccc(F)cc4)CC3)ccc21

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.82
HTR1A P08908 5/20 0.70
HTR2C P28335 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL466829 0.90 SIGMAR1 (1.00) SIGMAR1HTR1AHTR2C
SCHEMBL8948007 0.84 HTR1A (0.66) SIGMAR1HTR1AHTR2C
SCHEMBL8110473 0.83 SIGMAR1 (1.00) SIGMAR1HTR1AHTR2C
Hydrochloric Acid SCHEMBL9449919 0.82 HTR1A (0.98) SIGMAR1HTR1AHTR2C
SCHEMBL8114274 0.80 GRIN2B (0.60) SIGMAR1HTR1AHTR2C
SCHEMBL8958513 0.79 SIGMAR1 (0.53) SIGMAR1HTR1A
SCHEMBL8100660 0.78 SIGMAR1 (1.00) SIGMAR1HTR1AHTR2C
SCHEMBL8948030 0.77 SIGMAR1 (0.62) SIGMAR1HTR1AHTR2C
SCHEMBL9449853 0.76 HTR1A (0.86) SIGMAR1HTR1AHTR2C
SCHEMBL9449586 0.75 SIGMAR1 (0.69) SIGMAR1HTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688811-A PSYCHOLOGICAL DISORDERS; NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-11-18 US disclosed
US-5534511-A AFFINITY FOR SIGMA RECEPTORS, ANTIINFLAMMATORY, TREATMENT OF ARTHRITIS ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed