SCHEMBL8948018

SCHEMBL8948018

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)sc3cc(CCN4CCN(c5cccnc5)CC4)ccc32)CC1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.53
HTR2A P28223 5/20 0.49
HTR7 P34969 5/20 0.49
HTR2C P28335 4/20 0.49
HTR6 P50406 3/20 0.49
DRD4 P21917 2/20 0.48
DRD3 P35462 2/20 0.48
DRD2 P14416 1/20 0.46
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948011 0.91 HTR1A (0.60) HTR1AHTR2AHTR7HTR2CHTR6
SCHEMBL8947779 0.86 KDM4E (0.54) HTR1AHTR2AHTR7HTR2CSIGMAR1
SCHEMBL8948076 0.86 HTR1A (0.64) HTR1AHTR2AHTR7HTR2CHTR6
SCHEMBL8947985 0.86 KDM4E (0.58) HTR1AHTR2AHTR7HTR2CSIGMAR1
SCHEMBL8947935 0.83 HTR2A (0.59) HTR1AHTR2AHTR7HTR2CHTR6
SCHEMBL8947974 0.83 SIGMAR1 (0.64) HTR2AHTR7HTR2CHTR6SIGMAR1
SCHEMBL8948192 0.82 HTR1A (0.65) HTR1AHTR2AHTR7HTR2C
SCHEMBL8947762 0.81 HTR1A (0.66) HTR1AHTR2AHTR2CSIGMAR1
SCHEMBL8948007 0.80 HTR1A (0.66) HTR1AHTR2AHTR7HTR2CHTR6
SCHEMBL8948074 0.79 HTR1A (0.53) HTR1AHTR2AHTR7HTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed