SCHEMBL8948034

SCHEMBL8948034

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)sc3cc(O)ccc32)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.52
HTR2C P28335 2/20 0.52
HTR7 P34969 2/20 0.52
HTR6 P50406 2/20 0.52
SIGMAR1 Q99720 4/20 0.51
CNR2 P34972 2/20 0.51
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR1A P08908 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.50
DRD2 P14416 1/20 0.50
HPGD P15428 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD1 P21728 1/20 0.50
DRD4 P21917 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948121 0.87 HTR2A (0.57) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948150 0.87 HTR2A (0.55) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8947935 0.84 HTR2A (0.59) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948078 0.82 HTR2A (0.55) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8947974 0.82 SIGMAR1 (0.64) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948061 0.81 SIGMAR1 (0.52) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948051 0.81 HTR2A (0.55) HTR2AHTR2CHTR7HTR6ALDH1A1
SCHEMBL8948011 0.81 HTR1A (0.60) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL8948058 0.81 CNR2 (0.49) HTR2AHTR2CHTR7HTR6SIGMAR1
SCHEMBL11707845 0.81 KDM4E (0.58) HTR2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed