SCHEMBL8948150

SCHEMBL8948150

COc1ccc2c(c1)sc(=O)n2CCN1CCC(C(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.55
HTR2C P28335 2/20 0.55
DRD2 P14416 1/20 0.55
HSD11B1 P28845 3/20 0.51
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CNR2 P34972 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
HTT P42858 1/20 0.50
HTR7 P34969 1/20 0.48
HTR6 P50406 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948051 0.93 HTR2A (0.55) HTR2AHTR2CDRD2HSD11B1ALDH1A1
SCHEMBL8948034 0.87 HTR2A (0.52) HTR2AHTR2CDRD2ALDH1A1LMNA
SCHEMBL8947958 0.85 SMN1; SMN2 (0.55) LMNASMN1; SMN2
SCHEMBL8948121 0.83 HTR2A (0.57) HTR2AHTR2CDRD2ALDH1A1LMNA
SCHEMBL8947935 0.81 HTR2A (0.59) HTR2AHTR2CSIGMAR1HTR7HTR6
SCHEMBL8948192 0.81 HTR1A (0.65) HTR2AHTR2CHTR7
SCHEMBL8947963 0.81 SIGMAR1 (0.50) CNR2SIGMAR1
SCHEMBL8948061 0.80 SIGMAR1 (0.52) HTR2AHTR2CCNR2SIGMAR1HTR7
SCHEMBL8948000 0.80 HTR2A (0.50) HTR2AHTR2CDRD2SIGMAR1HTR7
SCHEMBL8948058 0.80 CNR2 (0.49) HTR2AHTR2CDRD2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed