SCHEMBL8948129

SCHEMBL8948129

O=c1[nH]c2ccc(CCCCN3CCN(c4cccc(C(F)(F)F)c4)CC3)cc2o1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.70
HTR2C P28335 3/20 0.70
DRD2 P14416 4/20 0.64
HTR2A P28223 2/20 0.63
SIGMAR1 Q99720 2/20 0.62
HTR7 P34969 5/20 0.55
SLC6A2 P23975 1/20 0.53
SLC6A3 Q01959 1/20 0.53
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
MAPT P10636 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP2C19 P33261 1/20 0.52
THPO P40225 1/20 0.52
MTOR P42345 1/20 0.52
BLM P54132 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10392901 0.97 DRD2 (0.67) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL10394028 0.83 DRD2 (0.62) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL8947948 0.82 HTR1A (1.00) HTR1AHTR2CDRD2HTR2ASIGMAR1
Hydrochloric Acid SCHEMBL7095759 0.80 HTR1A (0.54) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL10393591 0.79 HTR1A (0.59) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL10394830 0.79 HTR1A (0.65) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL6820733 0.78 DRD2 (1.00) HTR1AHTR2CDRD2HTR2ASIGMAR1
SCHEMBL9378627 0.78 SIGMAR1 (1.00) HTR1AHTR2CDRD2SIGMAR1HTR7
SCHEMBL4892696 0.77 HTR1A (0.64) HTR1AHTR2CDRD2HTR2AHTR7
SCHEMBL9595103 0.77 HTR1A (0.71) HTR1AHTR2CDRD2HTR2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0478446-A1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-04-01 EP claimed
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed