SCHEMBL8949083

SCHEMBL8949083

N=C(N)c1ccc(-c2ccc(NC3CCC(C(=O)O)CC3)nn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.43
ITGA2B P08514 8/20 0.43
HCAR3 P49019 3/20 0.42
PDK1 Q15118 1/20 0.41
ACHE P22303 1/20 0.41
DGAT1 O75907 1/20 0.41
KCNH2 Q12809 1/20 0.41
IL1B P01584 1/20 0.39
NLRP3 Q96P20 1/20 0.39
VCP P55072 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949075 1.00 ITGB3 (0.43) ITGB3ITGA2BHCAR3PDK1ACHE
SCHEMBL8949216 0.88 PDGFRB (0.43) ITGB3ITGA2BHCAR3PDK1ACHE
SCHEMBL8949224 0.88 PDGFRB (0.43) ITGB3ITGA2BHCAR3PDK1ACHE
SCHEMBL9571676 0.85 ITGB3 (0.46) ITGB3ITGA2BPDK1ACHEDGAT1
Hydrochloric Acid SCHEMBL8949349 0.81 ITGB3 (0.44) ITGB3ITGA2BHCAR3PDK1ACHE
SCHEMBL29818171 0.78 ACHE (0.52) PDK1ACHEIL1BNLRP3VCP
SCHEMBL8949306 0.76 ITGB3 (0.46) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8949315 0.76 ITGB3 (0.46) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL9252818 0.74 ADORA3 (0.41) ITGB3ITGA2BHCAR3DGAT1KCNH2
SCHEMBL9095484 0.74 MEN1 (0.61) ITGB3ITGA2BPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed