SCHEMBL8949442

SCHEMBL8949442

CCOC(=O)Cc1c(C)n(Cc2ccc(I)cc2)c2ccc(Br)cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 5/20 0.56
PTGS2 P35354 2/20 0.56
PTGES O14684 1/20 0.51
ALOX5 P09917 1/20 0.51
LMNA P02545 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
TSHR P16473 2/20 0.47
CYP2C19 P33261 2/20 0.47
PMP22 Q01453 2/20 0.47
MAPT P10636 2/20 0.47
PKM P14618 2/20 0.47
MEN1 O00255 1/20 0.47
RGS12 O14924 1/20 0.47
ALDH1A1 P00352 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47
GNAI1 P63096 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949489 0.93 PTGS2 (0.63) PLA2G2APTGS2PTGESALOX5LMNA
SCHEMBL8292054 0.89 PLA2G2A (0.70) PLA2G2APTGS2LMNAMAPTPKM
SCHEMBL8877441 0.84 PTGS2 (0.79) PLA2G2APTGS2LMNACYP1A2CYP3A4
SCHEMBL8292841 0.82 PLA2G2A (0.60) PLA2G2APTGS2LMNAMAPTPKM
SCHEMBL9286863 0.81 PLA2G2A (0.44) PLA2G2APTGS2PTGESALOX5LMNA
SCHEMBL8291608 0.81 PLA2G2A (0.60) PLA2G2APTGS2LMNATSHRMAPT
SCHEMBL9230125 0.79 PTGS2 (0.79) PLA2G2APTGS2PTGESALOX5LMNA
SCHEMBL8296317 0.79 LMNA (0.69) PLA2G2APTGS2LMNACYP1A2CYP3A4
SCHEMBL8291567 0.79 PLA2G2A (0.61) PLA2G2APTGS2LMNAMAPTPKM
SCHEMBL8292611 0.78 PLA2G2A (0.60) PLA2G2ALMNAMAPTPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037468-A1 N-BENZYL-3-INDOLEACETIC ACIDS AS CYCLOOXYGENASE-2-INHIBITORS AND ANTIINFLAMMATORY DRUGS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO disclosed
US-5510368-A INHIBITORS OF CYCLOOXYGENASE MERCK FROSST CANADA, INC. (CA) 1996-04-23 US disclosed