SCHEMBL8950955

SCHEMBL8950955

CCOC(=O)c1cc(C(N)=O)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.48
MMP13 P45452 1/20 0.48
CYP1A2 P05177 2/20 0.47
JMJD6 Q6NYC1 3/20 0.47
PIK3CA P42336 1/20 0.45
GABRP O00591 5/20 0.45
GABRD O14764 5/20 0.45
GABRA1 P14867 5/20 0.45
GABRB1 P18505 5/20 0.45
GABRG2 P18507 5/20 0.45
GABRB3 P28472 5/20 0.45
GABRA5 P31644 5/20 0.45
GABRA3 P34903 5/20 0.45
GABRA2 P47869 5/20 0.45
GABRB2 P47870 5/20 0.45
GABRA4 P48169 5/20 0.45
GABRE P78334 5/20 0.45
GABRA6 Q16445 5/20 0.45
GABRG1 Q8N1C3 5/20 0.45
GABRG3 Q99928 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL930636 0.89 JMJD6 (0.57) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL29466587 0.89 JMJD6 (0.57) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL581406 0.88 JMJD6 (0.57) CYP1A2JMJD6PIK3CANPC1RAB9A
SCHEMBL9297593 0.86 CYP1A2 (0.49) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL1920448 0.86 FTO (0.61) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL20963551 0.85 JMJD6 (0.44) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL29278613 0.85 JMJD6 (0.44) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL24604371 0.83 CYP1A2 (0.46) CYP1A2JMJD6PIK3CAGABRPGABRD
SCHEMBL3062909 0.81 ALDH1A1 (0.50) CYP1A2GABRPGABRDGABRA1GABRB1
Bromide SCHEMBL9298199 0.81 JMJD6 (0.44) CYP1A2JMJD6PIK3CAGABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed
WO-2010019204-A1 ANTIFUNGAL AGENTS MERCK SHARP & DOHME CORP. (US) 2010-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 MMP2 1070/4885MMP13 1527/4885CYP1A2 623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.