SCHEMBL8958326

SCHEMBL8958326

O=c1[nH]c2ccc(CCCCN3CCC(c4ccccc4)CC3)cc2s1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.67
HTR1A P08908 6/20 0.61
HTR2C P28335 6/20 0.61
MEN1 O00255 1/20 0.59
TP53 P04637 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
TSHR P16473 1/20 0.59
CYP2C19 P33261 1/20 0.59
KMT2A Q03164 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109930 0.92 HTR1A (0.69) SIGMAR1HTR1AHTR2CMEN1TP53
SCHEMBL8110695 0.86 SIGMAR1 (0.67) SIGMAR1HTR1AHTR2C
SCHEMBL8948027 0.84 HTR1A (0.57) SIGMAR1HTR1AHTR2CCYP1A2CYP3A4
SCHEMBL8947912 0.83 HTR1A (0.85) SIGMAR1HTR1AHTR2C
SCHEMBL8117008 0.80 SIGMAR1 (1.00) SIGMAR1HTR1AHTR2CMEN1TP53
SCHEMBL8109444 0.80 SIGMAR1 (0.58) SIGMAR1MEN1TP53CYP1A2CYP3A4
SCHEMBL8948040 0.80 HTR1A (0.61) SIGMAR1HTR1AHTR2C
SCHEMBL8948002 0.79 HTR1A (0.87) SIGMAR1HTR1AHTR2C
SCHEMBL7756727 0.79 HTR1A (0.64) HTR1AHTR2C
SCHEMBL8116065 0.78 HTR1A (0.67) SIGMAR1HTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534511-A AFFINITY FOR SIGMA RECEPTORS, ANTIINFLAMMATORY, TREATMENT OF ARTHRITIS ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed