SCHEMBL8959618

SCHEMBL8959618

C[C@@](N)(Cn1ccc2cc(Br)ccc21)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn1ccc2cc(Br)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
KRAS P01116 8/20 0.43
AR P10275 1/20 0.42
NTSR1 P30989 1/20 0.42
FABP4 P15090 2/20 0.38
FABP3 P05413 1/20 0.38
FABP2 P12104 1/20 0.38
FABP5 Q01469 1/20 0.38
HTR7 P34969 2/20 0.38
MCL1 Q07820 1/20 0.34
HDAC11 Q96DB2 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27340857 1.00 HTR2A (0.46) HTR2AHTR2CKRASARNTSR1
SCHEMBL27342171 0.87 HTR2C (0.45) HTR2AHTR2CFABP4MCL1HDAC8
SCHEMBL8959547 0.87 HTR2C (0.45) HTR2AHTR2CFABP4MCL1HDAC8
SCHEMBL8959588 0.86 HTR2A (0.46) HTR2AHTR2CKRASARHDAC8
SCHEMBL8959678 0.86 HTR2C (0.46) HTR2AHTR2CARFABP4HDAC8
SCHEMBL8959479 0.86 HTR2C (0.46) HTR2AHTR2CARFABP4HDAC8
SCHEMBL27524962 0.86 HTR2A (0.46) HTR2AHTR2CKRASARHDAC8
SCHEMBL8959608 0.82 HTR2A (0.45) HTR2AHTR2CARHDAC6HDAC1
SCHEMBL8959581 0.80 HTR2A (0.45) HTR2AHTR2CFABP4HTR7MCL1
SCHEMBL27528051 0.80 HTR2A (0.45) HTR2AHTR2CFABP4HTR7MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed