SCHEMBL8959581

SCHEMBL8959581

Cc1ccc2ccn(C[C@@](C)(N)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn3ccc4ccc(C)cc43)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.45
HTR2C P28335 2/20 0.45
HTR7 P34969 1/20 0.37
FABP4 P15090 1/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
APOBEC3A P31941 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
MCL1 Q07820 4/20 0.35
PRMT5 O14744 1/20 0.35
MTNR1A P48039 3/20 0.34
MTNR1B P49286 3/20 0.34
KMO O15229 2/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
SLC1A3 P43003 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27528051 1.00 HTR2A (0.45) HTR2AHTR2CHTR7FABP4KDM4E
SCHEMBL27342171 0.90 HTR2C (0.45) HTR2AHTR2CFABP4MCL1PRMT5
SCHEMBL8959547 0.90 HTR2C (0.45) HTR2AHTR2CFABP4MCL1PRMT5
SCHEMBL8959562 0.87 HTR2C (0.46) HTR2AHTR2CHTR7FABP4MTNR1A
SCHEMBL27356666 0.87 HTR2C (0.46) HTR2AHTR2CHTR7FABP4MTNR1A
SCHEMBL7997832 0.87 KMO (0.48) HTR2AHTR2CHTR7KDM4EALDH1A1
SCHEMBL8959608 0.83 HTR2A (0.45) HTR2AHTR2CMTNR1AMTNR1B
SCHEMBL8001823 0.82 MTNR1A (0.44) HTR2AHTR2CKDM4EALDH1A1POLB
SCHEMBL8959479 0.80 HTR2C (0.46) HTR2AHTR2CFABP4
SCHEMBL8959678 0.80 HTR2C (0.46) HTR2AHTR2CFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed