SCHEMBL8961083

SCHEMBL8961083

COc1ccccc1N1CCN(CCNc2nccc(C(N)=O)n2)CC1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.69
ADRA1D P25100 1/20 0.69
ADRA1B P35368 1/20 0.69
HTR1A P08908 6/20 0.61
DRD2 P14416 7/20 0.57
HTR2A P28223 4/20 0.57
HTR7 P34969 3/20 0.57
HTR6 P50406 3/20 0.57
DRD4 P21917 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9725708 0.95 ADRA1A (0.63) ADRA1AADRA1DADRA1BHTR1ADRD2
Fumaric Acid SCHEMBL9725713 0.95 ADRA1A (0.63) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9193895 0.88 ADRA1A (0.76) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9200004 0.87 ADRA1A (0.90) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9760100 0.86 HTR1A (0.64) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9759666 0.85 HTR1A (0.60) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9760272 0.84 DRD2 (0.67) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9759409 0.84 HTR1A (0.59) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9199195 0.83 ADRA1D (0.81) ADRA1AADRA1DADRA1BHTR1ADRD2
SCHEMBL9193482 0.82 ADRA1A (0.69) ADRA1AADRA1DADRA1BHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0435749-B1 Derivatives of 2-aminopyrimidine-4-carboxamide, their preparation and therapeutic use SYNTHELABO (FR) 1996-01-10 EP disclosed
EP-0435749-A1 Derivatives of 2-aminopyrimidine-4-carboxamide, their preparation and therapeutic use SYNTHELABO (FR) 1991-07-03 EP disclosed