SCHEMBL8963064

SCHEMBL8963064

FC(F)(F)Oc1ccc(C2CCC(CC[C@H]3CC[C@H](/C=C/Cl)CC3)CC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.37
ESR2 Q92731 3/20 0.36
KDM1A O60341 1/20 0.36
RCOR1 Q9UKL0 1/20 0.36
GRM2 Q14416 1/20 0.35
ESR1 P03372 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
DHODH Q02127 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC6A4 P31645 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963060 1.00 EPHX2 (0.37) EPHX2ESR2KDM1ARCOR1GRM2
SCHEMBL8962828 0.93 L3MBTL1 (0.38) EPHX2KDM1ARCOR1GRM2L3MBTL1
SCHEMBL8962816 0.93 L3MBTL1 (0.38) EPHX2KDM1ARCOR1GRM2L3MBTL1
SCHEMBL8963027 0.89 MEN1 (0.36) EPHX2KDM1ARCOR1GRM2L3MBTL1
SCHEMBL8962707 0.89 L3MBTL1 (0.41) EPHX2KDM1ARCOR1GRM2L3MBTL1
SCHEMBL8962715 0.89 L3MBTL1 (0.41) EPHX2KDM1ARCOR1GRM2L3MBTL1
SCHEMBL8963125 0.84 DRD2 (0.43) ESR2GRM2ESR1CYP3A4CYP2C9
SCHEMBL8963134 0.84 DRD2 (0.43) ESR2GRM2ESR1CYP3A4CYP2C9
SCHEMBL8458133 0.84 ESR2 (0.34) EPHX2ESR2KDM1ARCOR1GRM2
SCHEMBL8458130 0.84 ESR2 (0.34) EPHX2ESR2KDM1ARCOR1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed