SCHEMBL8964023

SCHEMBL8964023

COc1cccc(C=O)c1Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
MAPT P10636 5/20 0.54
LMNA P02545 5/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
PRMT1 Q99873 1/20 0.48
SRC P12931 1/20 0.48
MEN1 O00255 2/20 0.46
NPC1 O15118 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
TLR9 Q9NR96 1/20 0.46
NTSR1 P30989 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HSPB1 P04792 2/20 0.45
ERN1 O75460 2/20 0.45
HTR1A P08908 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1750713 0.83 TLR9 (0.48) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL27670279 0.81 LMNA (0.55) ALDH1A1MAPTLMNACYP1A2CYP2C9
SCHEMBL4387499 0.81 HTT (0.53) ALDH1A1MAPTLMNAMEN1NPC1
SCHEMBL8964117 0.80 ALDH1A1 (0.71) ALDH1A1MAPTLMNACYP1A2CYP2C9
SCHEMBL10434914 0.79 SRC (0.65) ALDH1A1LMNACYP1A2CYP2C9CYP2C19
SCHEMBL14451771 0.78 TLR9 (0.61) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL26936544 0.78 PTGS2 (0.59) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL8964199 0.77 ALDH1A1 (0.53) ALDH1A1MAPTLMNACYP1A2CYP2C9
SCHEMBL8964192 0.77 ALDH1A1 (0.50) ALDH1A1MAPTLMNACYP1A2CYP2C9
SCHEMBL4730558 0.77 PRMT1 (0.55) ALDH1A1MAPTLMNACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5525614-A TREATING VASCULAR RESTENOSIS, CNS DISORDERS WARNER-LAMBERT COMPANY (US) 1996-06-11 US disclosed
US-5489686-A CARDIOVASCULAR DISORDER, NERVOUS SYSTEM DISORDER, ANTIDIURETIC , PSYCHLOGICAL DISORDER, ANTIDEPRESSANTS WARNER-LAMBERT COMPANY (US) 1996-02-06 US disclosed
EP-0641326-A1 SUBSTITUTED 1,2,3,4-TETRAHYDROISOQUINOLINES WITH ANGIOTENSIN II RECEPTOR ANTAGONIST PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-03-08 EP disclosed
US-5350757-A Treatment of vascular restenosis, nervous system disorders and cognition enhancement WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed
WO-1993023378-A1 SUBSTITUTED 1,2,3,4-TETRAHYDROISOQUINOLINES WITH ANGIOTENSIN II RECEPTOR ANTAGONIST PROPERTIES WARNER-LAMBERT COMPANY (US) 1993-11-25 WO disclosed
US-5246943-A Substituted 1,2,3,4-tetahydroisoquinolines with angiotensin II receptor antagonist properties WARNER-LAMBERT COMPANY (US) 1993-09-21 US disclosed