SCHEMBL8964263

SCHEMBL8964263

Cc1ccc([C@H]2CC[C@H](/C=C/Cl)CC2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.40
OPRL1 P41146 1/20 0.40
CCR1 P32246 1/20 0.38
CCR5 P51681 1/20 0.38
CCR8 P51685 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
KDM5A P29375 1/20 0.36
PDE10A Q9Y233 5/20 0.35
NOTUM Q6P988 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAP4K4 O95819 1/20 0.33
DGAT1 O75907 1/20 0.33
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964261 1.00 OPRM1 (0.40) OPRM1OPRL1CCR1CCR5CCR8
SCHEMBL9542379 0.89 PDE10A (0.39) OPRM1OPRL1CCR1CCR5CCR8
SCHEMBL827646 0.84 CCR1 (0.52) OPRM1OPRL1CCR1CCR5CCR8
Ammonia Solution, Strong SCHEMBL17820158 0.82 CCR1 (0.50) OPRM1OPRL1CCR1CCR5CCR8
SCHEMBL8963382 0.80 PDE10A (0.37) PDE10ANOTUMNPC1RAB9ASMN1; SMN2
SCHEMBL9299861 0.80 DRD2 (0.39) DRD2DRD4KDM5APDE10ANOTUM
SCHEMBL9299863 0.80 DRD2 (0.39) DRD2DRD4KDM5APDE10ANOTUM
SCHEMBL8963379 0.80 PDE10A (0.37) PDE10ANOTUMNPC1RAB9ASMN1; SMN2
SCHEMBL8963386 0.78 PDE10A (0.33) PDE10A
SCHEMBL8963391 0.78 PDE10A (0.33) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed