SCHEMBL8965846

SCHEMBL8965846

CC(=O)c1ccc2c3c(ccc2c1)-c1ccc(C(=O)c2c(C)cccc2C)cc1C3c1ccc(O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
HTR7 P34969 2/20 0.36
HTR2B P41595 2/20 0.36
HSD17B1 P14061 2/20 0.34
CLK1 P49759 1/20 0.33
DYRK1A Q13627 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2A6 P11509 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
LMNA P02545 1/20 0.32
CHRNA1 P02708 1/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966077 0.77 MEN1 (0.43) ESR1ESR2ALDH1A1MAPTHPGD
SCHEMBL8966522 0.72 SRD5A2 (0.43) ESR1ESR2ALDH1A1MAPTHPGD
SCHEMBL8966115 0.72 ESR1 (0.39) ESR1ESR2ALDH1A1MAPTCLK1
SCHEMBL8965809 0.72 ESR1 (0.45) ESR1ESR2CLK1DYRK1ADYRK1B
SCHEMBL9571847 0.72 ESR1 (0.37) ESR1ESR2ALDH1A1MAPTHPGD
SCHEMBL9742252 0.68 ESR1 (0.45) ESR1ESR2
SCHEMBL8966236 0.68 ESR1 (0.53) ESR1ESR2ALDH1A1MAPTHPGD
SCHEMBL8966091 0.66 ESR1 (0.57) ESR1ESR2MAPTHPGDSMN1; SMN2
SCHEMBL8471075 0.65 ALDH1A1 (0.66) ALDH1A1MAPTHPGDCYP2A6MEN1
SCHEMBL7534293 0.65 ESR1 (0.47) ESR1ESR2ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0524742-B1 Benzo(a)fluorene compounds LILLY CO ELI (US) 1996-02-28 EP disclosed
EP-0524742-A2 Benzo(a)fluorene compounds ELI LILLY AND COMPANY (US) 1993-01-27 EP disclosed
US-5147880-A Estrogenic and antiestrogenic activity ELI LILLY AND COMPANY (US) 1992-09-15 US disclosed