SCHEMBL8966522

SCHEMBL8966522

O=C(c1ccccc1)c1ccc2c(c1)C(c1ccc(O)cc1)c1c-2ccc2cc(C(=O)c3ccc(Cl)cc3Cl)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.43
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 5/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
TP53 P04637 1/20 0.37
SERPINE1 P05121 1/20 0.36
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
CNR2 P34972 1/20 0.35
ABCC9 O60706 1/20 0.35
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966077 0.80 MEN1 (0.43) RAB9ANPC1MEN1KMT2AMAPT
SCHEMBL9571847 0.74 ESR1 (0.37) RAB9AMEN1KMT2AMAPTALDH1A1
SCHEMBL8965846 0.72 ESR1 (0.38) RAB9ANPC1MEN1KMT2AMAPT
SCHEMBL8966115 0.71 ESR1 (0.39) RAB9ANPC1MEN1KMT2AMAPT
SCHEMBL8965809 0.70 ESR1 (0.45) RAB9ANPC1MEN1KMT2AESR1
SCHEMBL610783 0.70 SRD5A2 (0.72) SRD5A2RAB9ANPC1MEN1KMT2A
SCHEMBL522683 0.69 SRD5A2 (0.74) SRD5A2RAB9ANPC1MEN1KMT2A
SCHEMBL29350361 0.69 SRD5A2 (0.74) SRD5A2RAB9ANPC1MEN1KMT2A
SCHEMBL17765409 0.68 ESR1 (0.43) RAB9AMAPTMAPK1TP53ESR1
SCHEMBL5068843 0.68 SRD5A2 (0.68) SRD5A2RAB9AMAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0524742-B1 Benzo(a)fluorene compounds LILLY CO ELI (US) 1996-02-28 EP disclosed
EP-0524742-A2 Benzo(a)fluorene compounds ELI LILLY AND COMPANY (US) 1993-01-27 EP disclosed
US-5147880-A Estrogenic and antiestrogenic activity ELI LILLY AND COMPANY (US) 1992-09-15 US disclosed