SCHEMBL8967277

SCHEMBL8967277

COC(=O)c1cc([N+](=O)[O-])c2ccccc2c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
HPGD P15428 3/20 0.54
KDM4E B2RXH2 2/20 0.54
NPSR1 Q6W5P4 1/20 0.54
AKR1C3 P42330 2/20 0.48
AKR1C2 P52895 2/20 0.48
AKR1C4 P17516 1/20 0.48
AKR1C1 Q04828 1/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
LMNA P02545 1/20 0.46
PDGFRB P09619 1/20 0.45
FGFR1 P11362 1/20 0.45
PDGFRA P16234 1/20 0.45
FLT1 P17948 1/20 0.45
FGFR3 P22607 1/20 0.45
KDR P35968 1/20 0.45
VCAM1 P19320 1/20 0.44
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443000 0.87 TSHR (0.49) ALDH1A1HPGDKDM4EAKR1C3AKR1C2
SCHEMBL5789105 0.79 AKR1C4 (0.55) ALDH1A1HPGDKDM4ENPSR1AKR1C3
SCHEMBL11026935 0.79 CTSB (0.53) ALDH1A1KDM4ENPSR1AKR1C3AKR1C2
SCHEMBL29272663 0.78 CASP6 (0.49) ALDH1A1KDM4EAKR1C3AKR1C2AKR1C4
SCHEMBL3741758 0.77 KDM4E (0.60) ALDH1A1HPGDKDM4ENPSR1MEN1
SCHEMBL8527632 0.76 HTT (0.42) ALDH1A1HPGDMEN1KMT2ADRD2
SCHEMBL8525974 0.76 PRMT5 (0.51) ALDH1A1HPGDKDM4ELMNADRD2
SCHEMBL2131809 0.76 KDM4E (0.59) ALDH1A1HPGDKDM4ENPSR1DRD2
SCHEMBL8416055 0.76 TDP1 (0.58) ALDH1A1HPGDKDM4EAKR1C3AKR1C2
SCHEMBL8966782 0.76 KDM4E (0.59) ALDH1A1HPGDKDM4ENPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585116-B1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LTD (GB) 1996-02-28 EP disclosed
US-5389684-A Treats disorder of central nervous system LILLY INDUSTRIES LIMITED (GB) 1995-02-14 US disclosed
EP-0585116-A1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LIMITED (GB) 1994-03-02 EP disclosed