SCHEMBL8967280

SCHEMBL8967280

CN(C)C(=CC=O)c1ccsc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
DAO P14920 1/20 0.42
HDAC1 Q13547 1/20 0.39
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
C5AR1 P21730 1/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
ALOX12 P18054 2/20 0.32
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GPR52 Q9Y2T5 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
KDR P35968 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24554795 0.76 CES2 (0.48) CES2CES1LCKFYNDAO
SCHEMBL2992590 0.74 LCK (0.41) CES2CES1LCKFYNDAO
SCHEMBL2992588 0.74 LCK (0.41) CES2CES1LCKFYNDAO
SCHEMBL28919959 0.73 ALDH1A1 (0.43) HPGDNPC1RAB9AALDH1A1MAPT
SCHEMBL9683260 0.73 ALDH1A1 (0.43) HPGDNPC1RAB9AALDH1A1MAPT
SCHEMBL9683262 0.73 ALDH1A1 (0.43) HPGDNPC1RAB9AALDH1A1MAPT
SCHEMBL22492769 0.72 HTT (0.46) HPGDALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL5242504 0.72 HTT (0.46) HPGDALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL29955578 0.72 CES2 (0.48) CES2CES1LCKFYNDAO
SCHEMBL4711102 0.72 CES2 (0.48) CES2CES1LCKFYNDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5543520-A ANTITUMOR AGENTS CIBA-GEIGY CORPORATION (US) 1996-08-06 US disclosed
EP-0672040-A1 FURTHER PYRIMIDINE DERIVATIVES AND THEIR PREPARATION Novartis AG (CH) 1995-09-20 EP disclosed
WO-1995009852-A1 FURTHER PYRIMIDINE DERIVATIVES AND THEIR PREPARATION CIBA-GEIGY AG (CH) 1995-04-13 WO disclosed