SCHEMBL8968361

SCHEMBL8968361

N#Cc1c(Cl)cc(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.54
TSHR P16473 2/20 0.48
MAPK1 P28482 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MERTK Q12866 2/20 0.40
TDP1 Q9NUW8 1/20 0.37
GPR35 Q9HC97 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TLR9 Q9NR96 1/20 0.37
GRIA1 P42261 2/20 0.37
GRIA2 P42262 2/20 0.37
GRIA3 P42263 2/20 0.37
GRIA4 P48058 2/20 0.37
GRM6 O15303 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11583829 0.84 GPR35 (0.56) VCAM1TSHRMAPK1ALDH1A1MERTK
SCHEMBL14825528 0.82 VCAM1 (0.47) VCAM1TSHRMAPK1ALDH1A1MERTK
SCHEMBL25329697 0.78 VCAM1 (0.47) VCAM1ALDH1A1MERTKTDP1NPC1
SCHEMBL952362 0.75 ALDH1A1 (0.45) TSHRMAPK1ALDH1A1GPR35MAPT
SCHEMBL5035508 0.75 ALDH1A1 (0.59) VCAM1TSHRALDH1A1TDP1GPR35
SCHEMBL2950121 0.74 VCAM1 (0.50) VCAM1TSHRMAPK1ALDH1A1MERTK
SCHEMBL31419521 0.74 VCAM1 (0.64) VCAM1TSHRMAPK1ALDH1A1TDP1
SCHEMBL11504122 0.74 VCAM1 (0.64) VCAM1TSHRMAPK1ALDH1A1TDP1
SCHEMBL21957846 0.74 VCAM1 (0.50) VCAM1TSHRMAPK1ALDH1A1MERTK
SCHEMBL6186068 0.74 ALDH1A1 (0.58) VCAM1TSHRMAPK1ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed