SCHEMBL8969006

SCHEMBL8969006

FC(F)(F)c1ccc2c(c1)N=C1C3CCC(C3)N1C2

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.52
HTR2C P28335 4/20 0.39
HTR2A P28223 3/20 0.39
HTR2B P41595 3/20 0.39
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
HTR6 P50406 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968874 0.90 CTSD (0.41) CTSDHTR2CHTR2AHTR2BALDH1A1
SCHEMBL8969065 0.84 CTSD (0.51) CTSDHTR2CHTR2AHTR2BCHRNB2
SCHEMBL8969263 0.80 CTSD (0.33) CTSDHTR2CHTR2AHTR2B
SCHEMBL8969499 0.80 CTSD (0.49) CTSDHTR2CHTR2AHTR2BHRH3
SCHEMBL8968949 0.77 OPRM1 (0.31) CTSD
SCHEMBL8969196 0.74 CTSD (0.49) CTSDHTR2CHTR2AHTR2BCHRNB2
SCHEMBL8969419 0.74
SCHEMBL8970140 0.74 CTSD (0.32) CTSD
SCHEMBL8969521 0.73 CTSD (0.40) CTSDHTR2CHTR2AHTR2BCHRNB2
SCHEMBL8968679 0.73 CTSD (0.47) CTSDHTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed