SCHEMBL8968679

SCHEMBL8968679

Clc1ccc2c(c1)N=C1C3CCCC(C3)N1C2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.47
ACHE P22303 2/20 0.41
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
KDM2B Q8NHM5 1/20 0.32
CTSG P08311 1/20 0.32
CMA1 P23946 1/20 0.32
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969499 0.92 CTSD (0.49) CTSDACHEHTR2AHTR2CHTR2B
SCHEMBL8969504 0.81 ACHE (0.40) CTSDACHEHTR2AHTR2CHTR2B
SCHEMBL8969466 0.81 CTSD (0.49) CTSDACHEHTR2AHTR2CHTR2B
SCHEMBL8968676 0.80 NOS1 (0.31) NOS1NOS2
SCHEMBL8968500 0.76 NOS1 (0.35) NOS1NOS2
SCHEMBL8969263 0.76 CTSD (0.33) CTSDHTR2AHTR2CHTR2BNOS3
SCHEMBL8970140 0.75 CTSD (0.32) CTSD
SCHEMBL8969006 0.73 CTSD (0.52) CTSDHTR2AHTR2CHTR2B
SCHEMBL8968949 0.73 OPRM1 (0.31) CTSD
SCHEMBL8969131 0.71 HRH3 (0.31) CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed