SCHEMBL8968874

SCHEMBL8968874

FC(F)(F)c1ccc2c(c1)CN1C(=N2)C2CCC1C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.41
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CHRNB2 P17787 2/20 0.32
CHRNA4 P43681 2/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
MEN1 O00255 2/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969006 0.90 CTSD (0.52) CTSDHTR2AHTR2CHTR2BHRH3
SCHEMBL8969521 0.84 CTSD (0.40) CTSDHTR2AHTR2CHTR2BNOS3
SCHEMBL8969764 0.80 PDE3B (0.34) HTR2AHTR2CHTR2BNOS3NOS1
SCHEMBL8969504 0.80 ACHE (0.40) CTSDHTR2AHTR2CHTR2BNOS3
SCHEMBL8969737 0.77 OPRM1 (0.31)
SCHEMBL8969544 0.74 CTSD (0.39) CTSDHTR2AHTR2CHTR2BNOS3
SCHEMBL8970140 0.74 CTSD (0.32) CTSD
SCHEMBL8969419 0.74
SCHEMBL8969065 0.73 CTSD (0.51) CTSDHTR2AHTR2CHTR2BCHRNB2
SCHEMBL8969499 0.72 CTSD (0.49) CTSDHTR2AHTR2CHTR2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed