SCHEMBL8969273

SCHEMBL8969273

CNC(=O)Oc1ccc2c(c1Cl)CN1C=CC=CC1=N2

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.38
MAOA P21397 4/20 0.38
ALDH1A1 P00352 2/20 0.30
PGR P06401 1/20 0.30
GAA P10253 1/20 0.30
PTGS1 P23219 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970442 0.78 KDM4E (0.30) ACHEMAOAALDH1A1
SCHEMBL8969417 0.78 MAOA (0.36) ACHEMAOA
SCHEMBL8969002 0.75 ACHE (0.39) ACHEALDH1A1PTGS1HSD17B10
SCHEMBL8969217 0.74 PDE3B (0.43) ALDH1A1HSD17B10
SCHEMBL8969665 0.72 ACHE (0.48) ACHEMAOAALDH1A1
SCHEMBL8969302 0.72 ACHE (0.50) ACHEMAOAALDH1A1
SCHEMBL8968414 0.71 ACHE (0.36) ACHEMAOA
SCHEMBL8968801 0.70 ACHE (0.36) ACHEMAOA
SCHEMBL8969986 0.70 MAOA (0.35) ACHEMAOAALDH1A1
SCHEMBL8968208 0.69 PDE3B (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed