SCHEMBL8970030

SCHEMBL8970030

Clc1cccc2c1CN1C(=N2)C2CCC1C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.50
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
BLM P54132 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
ACHE P22303 2/20 0.41
OPRM1 P35372 9/20 0.34
OPRL1 P41146 9/20 0.34
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
SLC18A3 Q16572 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
BCHE P06276 2/20 0.32
NOTUM Q6P988 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969496 0.84 HTR2C (0.36) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8968432 0.83 CTSD (0.48) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8969282 0.82 CTSD (0.34) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8969623 0.81 HTR2C (0.36) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8970388 0.81 CTSD (0.33) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8969666 0.81 CTSD (0.34) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8969131 0.80 HRH3 (0.31) CTSD
SCHEMBL8969508 0.80 PDE3B (0.33) CTSDLMNACYP1A2CYP3A4CYP2D6
SCHEMBL8969213 0.79 ACHE (0.40) CTSDACHEOPRM1OPRL1OPRD1
SCHEMBL8969017 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed