SCHEMBL8973399

SCHEMBL8973399

CC(=O)Nc1ccc2cc(S(=O)(=O)NCC(=O)O)ccc2c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
ALDH1A1 P00352 4/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
APEX1 P27695 1/20 0.54
KDM4E B2RXH2 3/20 0.50
KMT2A Q03164 2/20 0.50
BACE1 P56817 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MEN1 O00255 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GRIN2D O15399 1/20 0.49
GRIN3B O60391 1/20 0.49
GRIN1 Q05586 1/20 0.49
GRIN2A Q12879 1/20 0.49
GRIN2B Q13224 1/20 0.49
GRIN2C Q14957 1/20 0.49
GRIN3A Q8TCU5 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4824728 0.87 POLB (0.73) POLBALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4489812 0.83 LMNA (0.61) POLBALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL6438335 0.81 ALDH1A1 (0.69) ALDH1A1APEX1KDM4EKMT2ATDP1
SCHEMBL3905853 0.78 APEX1 (0.57) ALDH1A1APEX1KDM4EKMT2ATDP1
SCHEMBL948303 0.78 KDM4E (0.78) POLBALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL950400 0.77 SNCA (0.59) POLBSMN1; SMN2KDM4EKMT2AMEN1
SCHEMBL8425825 0.77 MAPT (0.60) POLBALDH1A1APEX1NPSR1
SCHEMBL8577441 0.76 MEN1 (0.68) ALDH1A1SMN1; SMN2KDM4EKMT2ATDP1
SCHEMBL4483600 0.76 LMNA (0.59) POLBALDH1A1SMN1; SMN2KDM4EKMT2A
Water SCHEMBL11035834 0.76 SNCA (0.58) POLBSMN1; SMN2KDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
EP-0305947-B1 HYDANTOIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS WELL AS THEIR USE MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-07-29 EP disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed