SCHEMBL8974563

SCHEMBL8974563

CS(=O)(=O)c1ccc(C2=CC(CO)C=C2c2ccc(F)cc2)cn1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.37
CDK9 P50750 1/20 0.36
PTGS1 P23219 3/20 0.35
PIK3CD O00329 1/20 0.35
PIP5K1C O60331 1/20 0.35
PIK3CB P42338 1/20 0.35
PI4KA P42356 1/20 0.35
PIK3CG P48736 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
HTR2A P28223 2/20 0.35
KCNH2 Q12809 2/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974451 0.88 CDK9 (0.37) PTGS2CDK9PTGS1PIK3CDPIP5K1C
SCHEMBL8974112 0.88 CDK9 (0.37) PTGS2CDK9PTGS1PIK3CDPIP5K1C
SCHEMBL8974185 0.87 CA1 (0.44) PTGS2PTGS1HTR2AKCNH2
SCHEMBL8974223 0.86 POLB (0.37) PTGS2PTGS1PI4KBKCNH2
SCHEMBL8973732 0.84 PTGS2 (0.40) PTGS2CDK9PTGS1PIK3CDPIP5K1C
SCHEMBL8973860 0.82 PTGS2 (0.35) PTGS2CDK9PTGS1PIK3CDPIP5K1C
SCHEMBL8974314 0.81 PTGS2 (0.55) PTGS2PTGS1KDM4ECYP1A2CYP3A4
SCHEMBL8974127 0.81 KDM4E (0.36) PTGS2CDK9PTGS1PIK3CDPIP5K1C
SCHEMBL8974505 0.80 PTGS2 (0.43) PTGS2CDK9PTGS1KDM4ENPC1
SCHEMBL8974426 0.79 POLQ (0.36) PTGS2CDK9PTGS1PIK3CDPIP5K1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed