SCHEMBL8974585

SCHEMBL8974585

COC(=O)C1(C(=O)OC)C=C(c2ccc(S(N)(=O)=O)cc2)C(c2ccc(C(F)(F)F)cn2)=C1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.46
CHRNA7 P36544 1/20 0.46
CA12 O43570 7/20 0.44
CA1 P00915 7/20 0.44
CA2 P00918 7/20 0.44
CA9 Q16790 7/20 0.44
MAPT P10636 1/20 0.42
CA4 P22748 4/20 0.40
CA7 P43166 4/20 0.40
TRPV1 Q8NER1 4/20 0.40
PTGS2 P35354 5/20 0.40
PTGS1 P23219 2/20 0.40
ADAMTS4 O75173 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CCR6 P51684 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973879 0.94 KIF11 (0.45) KIF11CHRNA7CA12CA1CA2
SCHEMBL8974421 0.92 PTGS2 (0.43) KIF11PTGS2PTGS1ADAMTS4
SCHEMBL8973781 0.88 KIF11 (0.59) KIF11CHRNA7CA12CA1CA2
SCHEMBL8974117 0.87 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8974407 0.86 PTGS2 (0.41) CA12CA1CA2CA9CA4
SCHEMBL8974327 0.85 KIF11 (0.50) KIF11CHRNA7CA12CA1CA2
SCHEMBL8974209 0.85 KIF11 (0.52) KIF11CHRNA7CA12CA1CA2
SCHEMBL8974757 0.84 CA2 (0.41) CA12CA1CA2CA9CA4
SCHEMBL8974073 0.83 KIF11 (0.50) KIF11CHRNA7CA12CA1CA2
SCHEMBL8973691 0.83 CA1 (0.43) KIF11CHRNA7CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed