SCHEMBL8974757

SCHEMBL8974757

COC(=O)C1(C(=O)OC)C=C(c2ccc(F)cc2)C(c2ccc(S(N)(=O)=O)cn2)=C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.41
CA9 Q16790 9/20 0.41
CA1 P00915 8/20 0.41
PTGS2 P35354 6/20 0.41
CA12 O43570 5/20 0.41
PTGS1 P23219 3/20 0.41
CA4 P22748 4/20 0.39
CA5A P35218 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
CA7 P43166 3/20 0.39
MAOA P21397 2/20 0.39
CA14 Q9ULX7 1/20 0.39
MAOB P27338 1/20 0.38
KIT P10721 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974407 0.93 PTGS2 (0.41) CA2CA9CA1PTGS2CA12
SCHEMBL8974101 0.91 PTGS2 (0.47) PTGS2PTGS1KIT
SCHEMBL8973879 0.88 KIF11 (0.45) CA2CA9CA1PTGS2CA12
SCHEMBL8974737 0.87 PTGS2 (0.51) CA2CA9CA1PTGS2CA12
SCHEMBL8974783 0.86 PTGS2 (0.47) PTGS2PTGS1KIT
SCHEMBL8974814 0.84 CA2 (0.43) CA2CA9CA1PTGS2PTGS1
SCHEMBL8974105 0.84 CA2 (0.45) CA2CA9CA1PTGS2PTGS1
SCHEMBL8974585 0.84 KIF11 (0.46) CA2CA9CA1PTGS2CA12
SCHEMBL8974701 0.81 PTGS2 (0.45) CA2CA9CA1PTGS2PTGS1
SCHEMBL8974702 0.81 PTGS2 (0.43) CA2CA9CA1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed