SCHEMBL8973691

SCHEMBL8973691

COC(=O)C1(C(=O)OC)C=C(c2ccc(S(N)(=O)=O)cc2)C(c2ccc(C(F)(F)F)nc2)=C1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.43
CA2 P00918 8/20 0.43
CA9 Q16790 7/20 0.43
CA12 O43570 6/20 0.43
CA14 Q9ULX7 4/20 0.43
KCNH2 Q12809 2/20 0.43
MAP4K4 O95819 1/20 0.43
PIK3CA P42336 1/20 0.43
MINK1 Q8N4C8 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
PTGS2 P35354 6/20 0.42
PTGS1 P23219 4/20 0.42
KIF11 P52732 1/20 0.40
LGMN Q99538 1/20 0.39
CA4 P22748 1/20 0.39
CA5A P35218 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117985 0.91 KCNH2 (0.51) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974835 0.87 CA1 (0.44) CA1CA2CA9CA12CA14
SCHEMBL8973781 0.85 KIF11 (0.59) CA1CA2CA9CA12CA14
SCHEMBL8973824 0.84 PTGS2 (0.46) CA1CA2CA9CA12CA14
SCHEMBL8974585 0.83 KIF11 (0.46) CA1CA2CA9CA12CA14
SCHEMBL8974771 0.82 KCNH2 (0.42) CA1CA2CA9CA12CA14
SCHEMBL8974393 0.82 KIF11 (0.46) CA1CA2CA9CA12KCNH2
SCHEMBL8973763 0.81 POLB (0.41) CA1CA2CA9CA12KIF11
SCHEMBL8974138 0.81 KIF11 (0.45) CA2CA9CA12KCNH2MAP4K4
SCHEMBL8973879 0.81 KIF11 (0.45) CA1CA2CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed