SCHEMBL8974737

SCHEMBL8974737

COC(=O)C1(C(=O)OC)C=C(c2ccc(F)cc2)C(c2ccc(S(N)(=O)=O)cc2)=C1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.51
PTGS1 P23219 8/20 0.51
CA1 P00915 7/20 0.50
CA2 P00918 7/20 0.50
CA9 Q16790 7/20 0.50
CA12 O43570 5/20 0.50
CA14 Q9ULX7 3/20 0.50
CA4 P22748 3/20 0.50
MAOA P21397 2/20 0.50
CA7 P43166 1/20 0.50
SOS1 Q07889 1/20 0.47
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974198 0.89 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8974407 0.87 PTGS2 (0.41) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974757 0.87 CA2 (0.41) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974660 0.86 CA1 (0.51) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973781 0.85 KIF11 (0.59) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974120 0.84 CA2 (0.49) CA1CA2CA9CA12CA14
SCHEMBL8974835 0.84 CA1 (0.44) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974231 0.82 CA9 (0.46) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973691 0.81 CA1 (0.43) PTGS2PTGS1CA1CA2CA9
SCHEMBL214628 0.80 PTGS2 (0.56) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed