SCHEMBL8974771

SCHEMBL8974771

COC(=O)C1C=C(c2ccc(S(N)(=O)=O)cc2)C(c2ccc(C(F)(F)F)nc2)=C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
MAP4K4 O95819 1/20 0.42
PIK3CA P42336 1/20 0.42
MINK1 Q8N4C8 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
CA1 P00915 8/20 0.42
CA2 P00918 8/20 0.42
CA9 Q16790 7/20 0.42
CA12 O43570 4/20 0.42
CA14 Q9ULX7 3/20 0.42
PTGS2 P35354 7/20 0.41
PTGS1 P23219 4/20 0.41
KIF11 P52732 1/20 0.40
CA4 P22748 1/20 0.38
CA5A P35218 1/20 0.38
CA5B Q9Y2D0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974639 0.87 CA1 (0.43) CA1CA2CA9CA12CA14
SCHEMBL8974564 0.87 PTGS2 (0.43) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974201 0.85 KIF11 (0.57) CA1CA2CA9CA12CA14
SCHEMBL8973885 0.84 KIF11 (0.46) CA1CA2CA9CA12CA14
SCHEMBL8974153 0.83 KIF11 (0.40) CA1CA2CA9CA12PTGS2
SCHEMBL8974254 0.83 PTGS2 (0.46) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8973691 0.82 CA1 (0.43) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974144 0.81 KIF11 (0.44) CA1CA2CA9CA12PTGS2
SCHEMBL8974270 0.81 KIF11 (0.46) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8973831 0.81 PTGS2 (0.50) CA1CA2CA9CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed